摘要
可乐定为-中枢降压药,经烯丙基化可生成新型心血管药物烯丙尼定。综述了可乐定和烯丙尼定的合成方法。
Clonidine is a kind of central antihypertensive drug and under-goes allylation to produce alinidine which is a new type of cardiovascular drug. The article dlscussed the synthetic methods of clonidine and alinidine.
出处
《河北化工》
1995年第2期43-46,共4页
Hebei Chemical Industry
关键词
可乐定
烯丙尼定
合成方法
降压药
心血管药物
clonidine,alinidine,synthesis,2,6-dichloroaniline, ethylene-diamine,2-nitro-chlorobenzene,dimethylamine,2,6-dichlorobenzoyl hydrazine