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抗炎药物的研制——环氧合酶的适度抑制策略 被引量:6

Innovation of anti-inflammatory drugs——strategy of moderate inhibition of cyclooxygenases
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作者 郭宗儒
机构地区 中国医学科学院
出处 《药学学报》 CAS CSCD 北大核心 2005年第11期967-969,共3页 Acta Pharmaceutica Sinica
关键词 抗炎药物 环氧合酶 适度抑制 anti-inflammatory drugs cyclooxygenases moderate inhibition
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参考文献13

  • 1Vane JR. Inhibition of prostaglandin synthesis as a mechanism of action for aspirin-like drugs [ J ]. Nat New Biol, 1971,231(25) :232 -235.
  • 2Xie WL, Chipman JG, Robertson DL, et al. Expression of a mitogen-responsive gene encoding prostaglandin synthase is regulated by mRNA splicing [ J]. Proc Nail Acad Sci USA, 1991,88(7) :2692 -2696.
  • 3Warner TD, Giuliano F, VojNovic I, et al. Nonsteroid drug selectivities for cyclo-oxygenases-1 rather than cyclooxygenase-2 are associated with gastrointestinal toxicity:A full in vitro analysis [ J ]. Proc Natl Acad Sci USA,1999,96 ( 13 ): 7563 - 7568.
  • 4FitzGerald GA. Cardiovascular pharmacology of nonselective nonsteroidal anti-inflammatory drugs and coxibs: clinical considerations [J]. Am J Cardiol, 2002,89(6A) :26D - 32D.
  • 5Khan KN, Paulson SK, VerBurg KM, et al.Pharmacology of cyclooxygenase-2 inhibition in the kidney[J]. Kidney Int, 2002,61(4) :1210 - 1219.
  • 6Waener TD, Mitchell JA. Cyclooxygenase-3 ( COX-3 ):filling in the gaps toward a COX continuum.? [ J ]. Proc Natl Acad Sci USA, 2002,99 (21): 13371 - 13373.
  • 7Vane JR. Biomedicine. Back to an aspirin a day? [J]Science, 2002,296 (5567) :474 - 475.
  • 8Tacconelli S, Capone ML, Patrignani P. Clinical pharmacology of novel selective COX-2 inhibitors [ J ].Curr Pharm Des, 2004,10(6) :589 -601.
  • 9Mitchell JA, Akarasereenont P, Thiemermann C, et al.Selectivity of nonsteroidal antiinflammatory drugs as inhibitors of constitutive and inducible cyclooxygenase[J]. Proc Natl Acad Sci USA, 1993,90(24) :11693 -11697.
  • 10de Leval X, Delarge J, Somers F, et al. Recent advances in inducible cyclooxygenase ( COX-2 ) inhibition [ J ].Curr Med Chem, 2000,7(10) :1041 -1062.

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