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噻唑环衍生物的合成 被引量:6

Synthesis of thiazole derivatives
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摘要 The target compounds were prepared from thioamides with a series of α-halogenated carbonylate compounds.Ethyl thiazole-5-carboxylate,4-(chloromethyl)-2-isopropylthiazole and 2-isopropyl-ethyl thiazole-5-carboxylate were obtained in yields of 60%,65% and 70% respectively. The target compounds were prepared from thioamides with a series of a - halogenated carbonylate compounds. Ethyl thiazole - 5 - carboxylate, 4 - (chloremethyl) - 2 - isopropylthiazole and 2 - isopropyl - ethyl thiazole - 5 - carboxylate were obtained in yields of 60% ,65% and 70% respectively.
出处 《化学研究与应用》 CAS CSCD 北大核心 2006年第2期186-188,共3页 Chemical Research and Application
关键词 噻唑衍生物 硫代酰胺 5-噻唑羧酸乙酯 4-氯甲基-2异丙基噻唑 2-异丙基-5-噻唑羧酸乙酯 thiazole derivatives thioamide ethyl thiazole - 5 - carboxylate 4 - (cldoromethyl) - 2 - isopropylthiazole 2 - isopropyl - ethyl thiazole - 5 - carboxyhte
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