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佳诺沙星的合成与抗菌作用 被引量:3

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摘要 佳诺沙星(garenoxacin,1)是第一个对革兰阳性菌、革兰阴性菌、厌氧菌以及非典型病原体具有优良广谱活性的6-去氟喹诺酮类抗菌药。本文分7-溴喹诺酮、二氢异吲哚和佳诺沙星三个部分归纳总结了它的合成方法。同时也概述了它对革兰阳性菌、革兰阴性菌、厌氧菌和衣原体、支原体等典型病原体的抗菌作用,并与其他氟喹诺酮类抗菌药进行比较。
出处 《国外医药(抗生素分册)》 CAS 2006年第3期100-104,共5页 World Notes on Antibiotics
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二级参考文献13

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