五元氮杂糖衍生物的实用有效合成方法

A Practical and Efficient Synthesis of Five-Membered Azasugar Derivatives

以D-葡萄糖为原料,经具有降冰片烷结构的双环缩醛中间体,合成了部分羟基保护的1-脱氧-D-氮杂阿拉伯糖衍生物,提供了一种合成五元氮杂糖衍生物的简便有效方法.

A practical and efficient synthesis of 1,4-dideoxy-l,4-imino-D-arabinol and its partially protected derivatives has been described via the key intermediate with a norbornane-like structure using D-glucose as a starting material.