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含噻二唑杂环的1，8-萘酰亚胺衍生物的合成与表征 被引量：2

Synthesis and characterization of the derivatives of 1,8-naphthalimides containing thiadiazole heterocycle
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摘要 以4-溴-1,8-萘酐为起始原料,通过硝化、亲电取代、氢化还原、关环和亚酰化反应,合成了目标产物3,4-[1,2,3]-噻二唑-N-丙基-1,8-萘酰亚胺和3,4-[1,2,3]-噻二唑-N-丁基-1,8-萘酰亚胺。 Two new derivatives of naphthalimides 3,4-[ 1,2, 3 ]-thiadiazole-N-propyl-1,8-naphthalimide and 3,4-[ 1,2,3]- thiadiazole-N-butyl-1, 8-naphthalimide were synthesized via nitration, nucleophilic substitution, hydrogenation, cyclization and imidafion of 4-bromo-naphthalic anhydride. The two compounds were characterized by IR, 1HNMR and elemental analysis.
作者 张业 覃雯 刘贤贤
机构地区 桂林师范高等专科学校化学与工程技术系
出处 《化学试剂》 CAS CSCD 北大核心 2008年第3期211-212,226,共3页 Chemical Reagents
基金 国家自然科学基金资助项目(20362002,20762001)
关键词 萘酰亚胺 噻二唑 杂环 合成 表征 naphthalimides thiadiazoles heterocycle synthesis characterization
分类号 O626 [理学—有机化学]
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参考文献8

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同被引文献23

  • 1高永建,张治军,薛群基.噻二唑衍生物的合成及摩擦学性能研究[J].化学研究,1998,9(1):35-38. 被引量：5
  • 2康茵,孙洪伟.含酯基的二巯基噻二唑二聚物的摩擦学性能[J].石油学报（石油加工）,2007,23(1):82-86. 被引量：24
  • 3康茵,孙洪伟,代振宇,龙军.噻二唑二聚物/丁氧基三乙二醇复合物的合成[J].石油炼制与化工,2007,38(2):57-60. 被引量：9
  • 4张庆春,邢锦娟,刘琳,钱建华.新型噻二唑衍生物在喷气燃料中的抗腐蚀性能研究[J].渤海大学学报（自然科学版）,2007,28(2):123-125. 被引量：6
  • 5NOVAK L, HOMYANSZKY G, ROHALY J, et al. Preparation of novel hexythiazox analogues [ J ] . Pestic. Sci. , 1997, 49 (1) :85-89.
  • 6VICINI P, GERONIKAKI A, INCERTI M, et al. 2-Heteroarylimino-5-benzylidene-4-thiazolidinones analogues of 2- thiazolylimino-5-benzylidene-4-thiazolidinones with antimicrobial activity : synthesis and structure-activity relationship[ J]. Bioorg. Med. Chem. ,2008,7(16) :3 714-3 724.
  • 7KIM D K, CHOI J H, AN Y J, et al. Synthesis and biological evaluation of 5- (pyridin-2-yl) thiazoles as transforming growth factor-β typel receptor kinase inhibitors [ J]. Bioorg. Med.Chem. Left. ,2008,6(18) :2 122-2 127.
  • 8ZHENG Ming-qiang, YIN Duan-zhi, QIAO Jin-ping, et al. Syntheses and evaluation of fluorinated benzothiazole anilines as potential tracers for/3-amyloid plaques in Alzheimer's disease[J]. J. Fluorine Chem. ,2008,3(29) :210-216.
  • 9PHILIPOVA T. Synthesis and application of fluorescent dyes on basis of 1, 8-naphthalic carboximides [ J ]. J. Prakt. Chem. , 1994,336(7) :587-590.
  • 10WOLARZ E, MORYSON H, BAUMAN D. Dichroic fluorescent dyes for guest-host' liquid crystal displays[J]. Displays, 1992,13(4) : 171-178.

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化学试剂
2008年 第3期

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