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截短侧耳素类衍生物及瑞他莫林的研究进展 被引量：5

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作者 游然 叶卉 宋婉玲 幸敏丽 潘腾洋 林克江 尤启东
机构地区 中国药科大学药学院
出处 《中南药学》 CAS 2009年第11期844-850,共7页 Central South Pharmacy
基金 中华医学会 江苏省教育厅资助(项目238号)
关键词 瑞他莫林 机制 药理活性 构效关系
分类号 R914 [医药卫生—药物化学]
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参考文献26

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同被引文献36

  • 1Li Qiang Fu,Xing Sheng Guo,Xin Liu,Hui Li He,Yu Ling Wang,Yu She Yang.Synthesis and antibacterial activity of C-2(S)-substituted pleuromutilin derivatives[J].Chinese Chemical Letters,2010,21(5):507-510. 被引量：5
  • 2王呈玉,图力古尔,李玉.侧耳属真菌系统分类研究概况[J].吉林农业大学学报,2006,28(2):158-163. 被引量：13
  • 3SCHLuNZEN F, ETAN E, FUCINI P, et al. Inhibition of Peptide Bond Formation by Pleuromutilins: The Structure of the 50s Ribosomal Subunit from Deinococcus Radiodurans in Complex with Tiamulin[J]. Molecular Microbiology, 2004, 54(5): 1287- 1294.
  • 4PRINGLE M, POEHLSGAARD J, VESTER B, et al. Mutations in Ribosomal Protein L3 and 23s Ribosomal Rna at the Peptidyl Transferase Centre are Associated with Reduced Susceptibility to Tiamulin in Brachyspira spp. Isolates[J]. Molecular Microbiology, 2004, 54(5): 1295-1306.
  • 5POULSEN S M, KARLSSON M, JOHANSSON L B, et al. The Pleuromutilin Drugs Tiamutin and Valnemulin Bind to the RNA at the Peptidyl Transferase Centre on the Ribosome[J]. Molecular Microbiology, 2001, 41(5): 1091-1099.
  • 6DORNHELM P, HOGENAUER G. The Effects of Tiamulin, a Semisynthetic Pleuromutilin Derivative, on Bacterial Polypepfide Chain Initiation[J]. Eur. J. Biochem. 1978, 91: 465-473.
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  • 8SCHUSTER I, FLESCHURZ C, HELM I. On the Interaction of a Lipophilic Drug with Different Sites of Rat-liver Microsomes Equilibrium Studies with a Substituted Pleuromutilin[J]. Eur J Biochem, 1975, 51: 511-519.
  • 9DAVIDOVICH C, BASHAN A, T AUERBACH-NEVO A, et al. Induced-fit Tightens Pleuromutilins Binding to Ribosomes and Remote Interactions Enable Their Selectivity[J]. PNAS, 2007, 104(11): 4291-4296.
  • 10LONG K S, POEHLSGAARD J, HANSEN L H, et al. Single 23S rRNA Mutations at the Ribosomal Peptidyl Transferase Centre Confer Resistance to Valnemulin and Other Antibiotics in Mycobacterium Smegrnatis by Perturbation of the Drug Binding Pocket[J]. Molecular Microbiology, 2009, 71(5): 1218-1227.

引证文献5

二级引证文献20

中南药学
2009年 第11期

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