不对称烷基化反应在药物及生物活性化合物合成中的应用
Application of asymmetric alkylation in the synthesis of pharmaceuticals and bioactive compounds
摘要
该文从合成光学活性化合物的3种手性诱导方式——手性源诱导的不对称反应、手性助剂诱导的不对称反应及不对称催化反应来介绍近年来不对称烷基化反应在药物及生物活性化合物合成中的应用。
Application of asymmetric alkylation in the synthesis of pharmaceuticals and bioactive compounds is reviewed categorized by chiral pool, chiral auxiliary and chiral catalysis.
出处
《中国药物化学杂志》
CAS
CSCD
2009年第6期463-475,497,共14页
Chinese Journal of Medicinal Chemistry
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