生物合理设计光系统Ⅱ抑制剂研究 (Ⅶ)──2-氰基-3-甲硫基-3-芳氨基丙烯酸乙酯的合成及其Hil反应抑制活性

Synthesis and Hill Inhibitory Activity of Ethyl\= 2Cyano3methylthio3arylaminoacrylates

合成了化合物２－氰基－３－甲硫基－３－芳氨基丙烯酸乙酯（２ａ＿２ｗ），产物结构通过１ＨＮＭＲ和元素分析证实，测定了所有化合物的Ｈｉｌ反应抑制活性．生物活性测定结果表明，部分化合物均表现出良好的抑制活性。

Based on our previous studies, the title compounds were designed and synthesized, all compounds have been confirmed by 1HNMR and elemental analysis. The Hill inhibitory activity of all titlecompounds were tested, and the bioassay results indicate that some of themshow a good inhibitory activity, the relationship between the structure andinhibitory activity was analyzed.