4KOMATSU T, YAMAZAKI H, SHIMADA N, et al. Involvement of microsomal cytochrome P450 and cytosolic thymidine phosphorylase in 5-fluorouracil formation from tegafur in human liver [J]. Clin Cancer Res, 2001, 7(3): 675 -681.
5YAMAZAKI H, KOMATSU T, TAKEMOTO K,, et al. Decreases in phenytoin hydroxylation activities catalysed by liver microsomal eytochrome P450 enzymes in phenytoin treated rats [J]. Drug Metab Dispos, 2001, 29(4 Pt 1): 427-434.
6日本药局方.16版[S].2011:1465-1466.
7IRINEL B, DANA M, AUREL T, et al. Determination of the 5-fluorouracil and Nl(2-furanidyl)uracil in the presence of tegafur by zero-crossing first derivative spectrometry [J]. J Pharm Biomed Anal, 2002, 30: 1371-1378.
8ROBERT D, EDWARD P, CHARLES H. The synthesis of 5-fluoroadenosines [J]. J Am Chem Soc, 1957, 79(16): 4559-4560.
9Shandong Newtime Pharmaceutical Co., LTD. An industrial synthesis method for adding fluorine: China, 103159746A [P]. 2013-06-19.
10GILLER S A, ZHUK R A, LIDAK M. Analogs of pyrimidine nucleosides. I. Nl-(alpha-furanidyl) derivatives of natural pyrimidine bases and their antimetabolities [J]. Dokl Akad Nauk SSSR, 1967, 176(2): 332-335.