Synthesis of some heteroaryl pyrazole derivatives and their biological activities 被引量：4

Synthesis of some heteroaryl pyrazole derivatives and their biological activities

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摘要 In order to search for novel fungicides with high activity, a series of heteroaryl pyrazoles were synthesized from 5-pyrazole formhydrazide. The structures of all new compounds were confirmed by spectroscopic methods and microanalyses. Preliminary bioassays indicated that some compounds showed fungicidal activity against Puccinia tritinia and PGR activity as well. In order to search for novel fungicides with high activity, a series of heteroaryl pyrazoles were synthesized from 5-pyrazole formhydrazide. The structures of all new compounds were confirmed by spectroscopic methods and microanalyses. Preliminary bioassays indicated that some compounds showed fungicidal activity against Puccinia tritinia and PGR activity as well.

作者陈寒松李正名

机构地区 State Key Laboratory of Elemento-Organic Chemistry

出处《Chinese Journal of Chemistry》 SCIE CAS CSCD 2000年第4期596-602,共7页 中国化学（英文版）

基金 Project (No. 29832050) supported by the National Natural Science Foundation of China.

关键词 5-(Substituted-pyrazol-5′-yl)-1 3 4-thiadiazole 5-(substituted-pyrazol-5′-yl)-l 2 4-triazole 5-(substituted-pyrazol-5′-yl)-1 3 4-oxadiazole fungicidal activity PGR activity 5-(Substituted-pyrazol-5′-yl)-1, 3,4-thiadiazole 5-(substituted-pyrazol-5′-yl)-l,2,4-triazole 5-(substituted-pyrazol-5′-yl)-1,3,4-oxadiazole fungicidal activity PGR activity

分类号 O626 [理学—有机化学]

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Chinese Journal of Chemistry

2000年第4期

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Synthesis of some heteroaryl pyrazole derivatives and their biological activities 被引量：4

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