摘要
2010年11月15日,美国FDA批准了日本卫材公司研发用于治疗转移性乳腺癌的新药甲磺酸艾日布林(efibulinmesylate,商品名Halaven)上市,本品是一种微管抑制剂,其抗癌作用机制与紫杉醇基本相同。其分子式为C40H59NO11·CH4O3S,分子量为826.0(游离碱为729.9)。
出处
《中国药学杂志》
CAS
CSCD
北大核心
2011年第23期1855-1856,共2页
Chinese Pharmaceutical Journal
参考文献4
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1FDA. Label approved on 11/15/2010 for HALAVEN, NDA no. 201532 [ EB/OL]. http://www, accessdata.fda, gov/drugsatfda docs/label/2010/2015321bl, pdf.
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4JAVIER C, ALBERTO J M, STEFAN G. Eribulin rnesylate, a novel microtubule inhibitor in the treatment of breast cancer [ J ]. Cancer Treat Rev, 2011, 22(10) :1-12.
同被引文献10
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