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根皮素乙酰阿魏酸酯的合成及抗氧化活性研究 被引量:12

Synthesis and Antioxidant Activity of Phloretin Acetylferulic Acid Esters
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摘要 以阿魏酸和根皮素为原料,合成了三种根皮素乙酰阿魏酸酯,采用IR、1H NMR、13C NMR和HPLC-MS对其结构进行表征。并测定根皮素及其酯的还原能力、清除DPPH自由基及.OH自由基能力,结果表明根皮素乙酰阿魏酸酯的抗氧化活性显著优于根皮素。 Three new compounds were firstly synthesized by ferulic acid and phloretin. The target compound was charac- terized by IR,IH NMR,13C NMR and HPLC-MS,respectively. Reducing POwer,DPPH and · OH radical scavenging as- says were carried out to evaluate the antioxidant and free radical scavenging abilities of phloretin and its esters. The re- suits showed that the antioxidant and free radical scavenging abilities of phloretin acetylferulic acid esters were stronger than that of phloretin.
出处 《天然产物研究与开发》 CAS CSCD 北大核心 2012年第3期316-320,共5页 Natural Product Research and Development
基金 国家自然科学基金(20962014)
关键词 根皮素 阿魏酸 酯化 合成 抗氧化 phloretin femlic acid esterification antioxidant activity synthesis
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