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Design, Synthesis and Biological Activities of Novel Benzoyl Hydrazines Containing Pyrazole 被引量:4

Design, Synthesis and Biological Activities of Novel Benzoyl Hydrazines Containing Pyrazole
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摘要 In search of environmentally benign compounds with high biological activity, low toxicity and low resistance, 8 novel benzoyl hydrazines containing pyrazole were designed and synthesized. All compounds were characterized by I H NMR spectra and HRMS. The preliminary results of biological activity assessment indicated that most of title compounds exhibited certain insecticidal activities against M),thimna separata Walker at 200 mg L-1 but excellent fungicidal activities against six fungus at 50 mg L-1, which were better than the control. In search of environmentally benign compounds with high biological activity, low toxicity and low resistance, 8 novel benzoyl hydrazines containing pyrazole were designed and synthesized. All compounds were characterized by I H NMR spectra and HRMS. The preliminary results of biological activity assessment indicated that most of title compounds exhibited certain insecticidal activities against M),thimna separata Walker at 200 mg L-1 but excellent fungicidal activities against six fungus at 50 mg L-1, which were better than the control.
出处 《Chinese Journal of Chemistry》 SCIE CAS CSCD 2012年第4期919-923,共5页 中国化学(英文版)
关键词 benzoyl hydrazines PYRAZOLE SYNTHESIS insecticidal activities fungicidal activities benzoyl hydrazines, pyrazole, synthesis, insecticidal activities, fungicidal activities
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