α-芳氨基乙酰芳胺的合成及除草活性

Synthesis and herbicidal activity of Q-aromaticaminoacetic aromaticamine

对α-芳氨基乙酰芳胺的合成路线作了小结，优化了传统反应条件，发现加入碘化钾作为催化剂后，反应时间短，条件温和，收率高，在优化条件下合成了11个α-芳氨基乙酰芳胺；对产物进行了1HNMR和MS表征；除草活性测试表明产物对双子叶植物的根有较好的抑制作用．

The synthesis and herbicidal activity of eleven α-aromaticaminoacetic aromaticamines are reported. Adding KI as a catalyst results in the mild reaction condition and good yield in the synthesis. The structures of these title compounds are characterized by H NMR and MS.