Efficient Regioselective Synthesis of 3-1odoindole N-Carboximidamides and N-Carboximidoates by a Sequential Aza-Wittig/Iodine Induced Cyclization

Efficient Regioselective Synthesis of 3-1odoindole N-Carboximidamides and N-Carboximidoates by a Sequential Aza-Wittig/Iodine Induced Cyclization

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摘要 3-Iodoindole N-carboximidamides and N-carboximidoates 4 were prepared regioselectively via a sequential aza-Wittig/iodine induced cyclization, starting from easily accessible 2-alkynylphenyl iminophosphorane, isocyanates, various nucleophiles and iodine. 3-Iodoindole N-carboximidamides and N-carboximidoates 4 were prepared regioselectively via a sequential aza-Wittig/iodine induced cyclization, starting from easily accessible 2-alkynylphenyl iminophosphorane, isocyanates, various nucleophiles and iodine.

作者聂熠博段专丁明武

机构地区 Key Laboratory of Pesticide&Chemical Biology of Ministry of Education

出处《Chinese Journal of Chemistry》 SCIE CAS CSCD 2012年第8期1807-1812,共6页 中国化学（英文版）

关键词 indole aza-Wittig reaction IODINE CYCLIZATION IMINOPHOSPHORANE indole, aza-Wittig reaction, iodine, cyclization, iminophosphorane

分类号 TQ655 [化学工程—精细化工] O623.712 [理学—有机化学]

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Chinese Journal of Chemistry

2012年第8期

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Efficient Regioselective Synthesis of 3-1odoindole N-Carboximidamides and N-Carboximidoates by a Sequential Aza-Wittig/Iodine Induced Cyclization

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