2HUANG WS,METCALF CA,SUNDARAMOORTHI R,et al.Discovery of 3-[2-(Imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-N-{4-[(4-methylpiperazin-1-yl)-methyl]-3-(trifluoromethyl)phenyl}benzamide (AP24534),a potent,orally active pan-inhibitor of breakpoint cluster region-abelson (BCR-ABL) kinase including the T315I gatekeeper mutant[J].J Med Chem,2010,53:4701-4719.
3ZUPAN M,POLLAK A.Fluorination with xenon difluoride.Reaction with halogenated hydrocarbons[J].J Fluor Chem,1976,8(3):275-278.