摘要
12H-Dibenzo d,g 1,3 dioxocin-6-carboxylic acid is a patented herbicide (US4976770)With good pre-and post-emergence activity on dicot weeds and sedges. Structure activity studies were initiated with the goal of discovering more synthetically accessible analogs with improved unit activity and crop-weed selectivity.An improved procedure to prepare the lead compound was developed.Analogs were prepared in which both the tricyclic core and the carboxylic acid function were varied.The synthesis and screening results of these analogs will be presented.
12H-Dibenzo d,g 1,3 dioxocin-6-carboxylic acid is a patented herbicide (US4976770)With good pre-and post-emergence activity on dicot weeds and sedges. Structure activity studies were initiated with the goal of discovering more synthetically accessible analogs with improved unit activity and crop-weed selectivity.An improved procedure to prepare the lead compound was developed.Analogs were prepared in which both the tricyclic core and the carboxylic acid function were varied.The synthesis and screening results of these analogs will be presented.
出处
《浙江化工》
CAS
2000年第C00期26-26,共1页
Zhejiang Chemical Industry
关键词
二氧环辛烷
羧酸类
三环化合物
除草活性
除草剂
12H-Dibenzo d,g dioxocin-6-carboxylic acid,herbicide,structure and activity