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四唑酰草胺合成方法述评 被引量:1

A Review of Synthetic Methods of Fentrazamide
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摘要 总结了文献报道的四唑酰草胺及其中间体的合成工艺路线和具体的合成方法。四唑酰草胺由关键中间体苯基四唑啉酮进行多步反应得到,主要有2条工艺路线。 The synthetic method and detailed process of fentrazamide and its intermediates reported in the literature were summarized. Fentrazamide was synthesized via several reaction steps from phenyl substituted tetrazolones. There were mainly two different processes to synthesis fentrazamide.
出处 《农药》 CAS CSCD 北大核心 2013年第10期776-777,共2页 Agrochemicals
基金 十二五”国家科技支撑计划项目(2011BAE06B00) 国家重点基础研究计划(973计划)项目(2012CB724501)
关键词 四唑酰草胺 工艺路线 合成方法 fentrazamide process synthetic method
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参考文献5

  • 1REINHARD L, UWE S, CARL C. Process for Preparing l-Aryl- 4-carbamoyl-tetrazoliones: US, 5874586[P]. 1999-02-23.
  • 2GOTO T, ITO S, WATANABE Y, et al. Herbicidal Tetrazolinones: EP, 0672663[P]. 1995-09-25.
  • 3AKIHIKO Y, YUKIYOSHI W, SHIN-ICHI N. Process for the Production of 1-Substituted-5-(4H)-tetrazolinones: US, 5530135[P]. 1996-06-25.
  • 4LANTZSCH R, STELZER U. Process for the Production of 1-Aryl-4-carbamoyl-tetrazolinones. EP, 0764642[P]. 1997-03-26.
  • 5兰施R,施特尔策U.卡泽C.1-芳基-4-氨基甲酰基四唑啉酮的制备:ZL.96120142[P].2001-01-10.

同被引文献43

  • 1夏成才,程冬萍,于文博,颜继忠.第四代头孢研究进展及合成综述[J].应用化工,2005,34(3):137-140. 被引量:14
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  • 4AL-HOURANI B J, SHARMA S K, MANE J Y, et ol. Synthesis and Evaluation of 1,5-Diaryl-substituted Tetrazoles as NovelSelective Cyclooxygenase-2 (COX-2)Inhibitors[J]. Bioorganic & Medicinal Chemistry Letters, 2011, 21(6): 1823-1826.
  • 5WANASKI S, COLLINS S, K1NCAID J. Arylsulfonamide Derivatives as Sodium-potassium-chloride Cotransporter Inhibitors and Their Preparation, Compositions, and Methods of Use: WO, 2012018635[P]. 2012-02-09.
  • 6PRONSKII L F, ABRAZHANOVA E A, SEVAST'YANOV V N. Synthesis of 5-(Sulfonylamido)-1-aryltetrazole[J]. Voprosy Khimii i Khimicheskoi Tekhnologii, 1974, 33: 10-14.
  • 7TRECANT C, DLUBALA A, GEORGE P, et ol. Synthesis and Biological Evaluation of Analogues of M6G[J]. European Journal of Medicinal Chemistry, 2011, 46(9): 4035-4041.
  • 8BURGOS-LEPLEY C E, THOMPSON L R, KNEEN C O, et 01. Carboxylate Bioisosteres of Gabapentin[J]. Bioorganic & Medicinal Chemistry Letters, 2006, 16(9): 2333-2336.
  • 9SCHWARZ J B, COLBRY N L, ZHU Z, et 01. Carboxylate Bioisosteres ofPregabalin [J]. Bioorganic & Medicinal ChemistryLetters, 2006, 16(13): 3559-3563.
  • 10YUAN H, SILVERMAN R B. Structural Modifications of (1S,3S)- 3-Amino-4-difluoromethylene Cyclopentanecarboxylic Acid, a Potent Irreversible Inhibitor of GABA Aminotransferase [J]. Bioorganic & Medicinal Chemistry Letters, 2007,17(6): 1651-1654.

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