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血管紧张素Ⅱ受体拮抗剂 被引量:4

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摘要 血管紧张素Ⅱ(AⅡ)是R-A系统的生物活性中心。本文概述了AⅡ的生理活性、肽类AⅡ受体拮抗剂、非肽类Ⅰ型AⅡ受体拮抗剂DuP753和Ⅱ型AⅡ受体拮抗剂EXP655.DuP753对高肾素高血压和卡托普利有相当的降压效果,未见咳嗽副作用,对低肾素高血压无效。
作者 蒋伯诚
机构地区 常州制药厂
出处 《药学进展》 CAS 北大核心 1993年第1期4-10,共7页 Progress in Pharmaceutical Sciences
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