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他扎罗汀(乙炔维甲酸)的研究进展 被引量:23

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摘要 他扎罗汀是第一个根据受体选择性而研制的第三代维甲酸类药物 ,选择性地结合维甲酸受体 (RAR) ,但不结合维甲酸X受体 (RXR) ,调节银屑病的三个病理特征。他扎罗汀体内代谢迅速 ,系统吸收有限 ,无组织蓄积 ,可单独或联合治疗银屑病、痤疮、鱼鳞病、Darier病等 ,不良反应少、小 ,临床应用前景广阔。
出处 《中国皮肤性病学杂志》 CAS 北大核心 2001年第3期200-202,共3页 The Chinese Journal of Dermatovenereology
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