7-硝基-5-甲氧基-3-氨基-1.3-二氢-2酮吲哚的合成

Synthesis of 7-nitro-5-methoxy-3-ramino-1,3-dihydro - 2-one Indole

本文报导以对茴香胺为原料,通过硝化、酰化、环化、缩合和还原合成标题化合物。该化合物是一种新型吲哚醌衍生物,可用作合成二氢吲哚酮的酰胺衍生物的前体,其合成方法尚未见报导。

This paper describes the synthesis of new indole derivatives(Ⅵ ) dy the several steps reactions of nitration, acylation, cyciization, condensation, and reduction from 4-amidoanjsle, The title compound have not been nitherto reported in literature. It is important intermediate of preparation of 3-amide-2-one indole.