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4-(吡啶-2-甲氧基)-5,6,7,8-四氢萘酚-1-胺的合成

Synthesis of 4-(Pyridin-2-methoxy)-5,6,7,8-tetrahydro-1-aminonaphthol
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摘要 以α-萘酚为起始原料,经过5步反应得到4-(吡啶-2-甲氧基)-5,6,7,8-四氢萘酚-1-胺,总收率为27%。该制备工艺原料易得、反应条件温和、后处理简单,适合实验室的小规模制备。 4-(Pyridin-2-methoxy)-5,6,7,8-tetrahydro-l-aminonaphthol was synthesized in five-steps using α- naphthol as the starting material, and the overall yield was 27%. The advantages of this improved process included lower prices of commercial starting materials, mild reaction conditions, and suitable for bench-scale production.
出处 《精细化工中间体》 CAS 2015年第1期50-52,56,共4页 Fine Chemical Intermediates
关键词 4-(吡啶-2-甲氧基)-5 6 7 8-四氢萘酚-1-胺 Α-萘酚 4-(pyridin-2-methoxy)-5,6,7,8-tetrahydro-l-aminonaphthol α- naphthol synthesized
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