摘要
A novel copper-catalyzed direct C–N formation reaction of simple arenes with cheap and pharmacological saccharin derivatives under relatively mild conditions was developed with arenes as limiting reagents.This work provided a new method for oxidative coupling of aromatic C(sp2)–H bonds and N–H bonds.
A novel copper-catalyzed direct C-N formation reaction of simple arenes with cheap and pharmacological saccharin deriva- tives under relatively mild conditions was developed with arenes as limiting reagents. This work provided a new method for oxidative coupling of aromatic C(sp2)-H bonds and N-H bonds.
基金
financially supported by the National Natural Science Foundation of China(21172033,21372041,21302017)