摘要
与简单 aroyl 一种肺结核特效药联合吲哚的反应的崭新的钯 / 铜 cocatalyzed 在氧气的条件下面被开发了。aroyl 一种肺结核特效药的一个范围经历了钯 / 铜 cocatalyzed 有对在 dimethyl sulfoxide 和 nitromethane 的 1:1 混合物的空气开放的吲哚的氧化 arylation 节制给在结构上多样的 2-arylindoles 或 3-arylindoles 在里面到好收益。反应很好容忍许多功能的组象 alkoxy 那样，光圈，酉旨。
An unprecedented palladium/copper cocatalyzed coupling reaction of indoles with simple aroyl hydrazides has been developed under aerobic conditions. A range of aroyl hydrazides underwent palladium/copper cocatalyzed oxidative arylation with indoles open to air in a 1：1 mixture of dimethyl sulfoxide and nitromethane to give structurally diverse 2-arylindoles or 3-arylindoles in moderate to good yields. The reaction well tolerates a wide variety of functional groups such as alkoxy, halo, ester.
