摘要
银杏内酯类成分作为银杏叶的重要活性成分,具有较高的药用价值,在临床上应用广泛。该文综述了近年来国内外学者关于银杏内酯类化学成分、构效关系、分析方法、生物活性及药代(ADME)特征等方面的研究成果,为更加深入地开发利用银杏内酯提供参考依据。
Ginkgo terpene lactones,as an important active ingredient from Ginkgo leaves,has high medicinal values and has been widely used in clinics. This article would review the researches both at home and abroad,including chemical composition,structureactivity relationship,analytical methods,pharmacological effects,pharmacokinetic characteristics,and so on,providing a reference for further development and utilization of ginkgo terpene lactones.
作者
耿婷
申文雯
王佳佳
黄文哲
王振中
萧伟
GENG Ting;SHEN Wen-wen;WANG Jia-jia;HUANG Wen-zhe;WANG Zhen-zhong;XIAO Wei(Jiangsu Kaaion Parmaceutical Co. , Ltd. , Lianyungang 222001, China;State Key Laboratory of New-tech for Chinese Medicine Pharmaceutical Process, Lianyungang 222001, China)
出处
《中国中药杂志》
CAS
CSCD
北大核心
2018年第7期1384-1391,共8页
China Journal of Chinese Materia Medica
基金
国家“重大新药创制”科技重大专项(2013ZX09402203)
关键词
银杏内酯
化学成分
构效关系
分析方法
生物活性
药代(ADME)
ginkgo terpene lactones
chemical composition
structure-activity relationship
analytical methods
pharmacological effects
pharmacokinetic characteristics (ADME)