摘要
青蒿为常用中药,主要含有倍半萜、二萜、黄酮、苯丙酸、香豆素、黄酮和挥发油等多种类型化学成分,具有抗疟疾、抗肿瘤、抑菌杀虫、解热抗炎、免疫调节等药理活性。显著的抗疟活性使青蒿较早就用于疟疾的治疗。对近年来有关青蒿的化学成分及药理活性进行综述,以期为其进一步的开发与合理利用提供参考。
As a commonly used Chinese materia medica, Artemisia annua mainly contains sesquiterpenoids, diterpenes, phenylpropionic acids, coumarins, flavonoids, volatile oil, and other chemical compositions. Its pharmacological activities are anti-malaria, anti-tumor, anti-microbial, anti-parasitic, antipyretic, anti-inflammatory, immunoregulation and so on. The significantly anti-malarial activity has led to its earlier use in the treatment of malaria. In this paper, the chemical constituents and pharmacological activities of A. annua in recent years are reviewed in order to provide a reference for the further development and rational utilization of this plant resource.
作者
李海波
秦大鹏
葛雯
王振中
曹亮
肖伟
于洋
姚新生
LI Hai-bo;QIN Da-peng;GE Wen;WANG Zhen-zhong;CAO Liang;XIAO Wei;YU Yang;YAO Xin-sheng(Kanion Pharmaceutical Co., Ltd., Lianyungang 222001, China;State Key Laboratory of New-tech for Chinese Medicine Pharmaceutical Process, Lianyungang 222001, China;Key Laboratory for New Technique Research ofTCM Extraction and Purification, Lianyungang 222047, China;Institute of Traditional Chinese Medicine and Natural Products, Jinan University, Guangzhou 510632, China;Zhejiang Pharmaceutical College, Ningbo 315100, China)
出处
《中草药》
CAS
CSCD
北大核心
2019年第14期3461-3470,共10页
Chinese Traditional and Herbal Drugs
基金
国家自然科学基金重点项目(81630097)
热毒宁注射液标准化建设(ZYBZH-C-JS-31)
桂枝茯苓胶囊标准化建设(ZYBZH-C-JS-28)
关键词
青蒿
倍半萜类
黄酮类
抗疟疾
解热
抗炎
Artemisia annua L.
sesquiterpenoids
flavonoids
antimalaria activity
antipyretic effect
anti-inflammatory activity