摘要
发展了一种高效实用的氨化咪唑[1,2-α]吡啶类化合物的方法.值得注意的是,该反应无需任何金属催化剂参与.在中等至高收率下,成功得到了带有多样取代基的产物.
A highly efficient and practical amination protocol for imidazo[1,2-α]pyridines using heteroaromatic amines was developed.Notably,the transformation proceeds without the need for any metal catalyst.Isolation of products bearing diverse substituents was achieved in moderate to high yields.
作者
孙一平
陈德茂
何玲
王祖利
Sun Yiping;Chen Demao;He Ling;Wang Zuli(State Key Laboratory of Solid Lubrication,Lanzhou Institute of Chemical Physics,Chinese Academy of Sciences,Lanzhou 730000;College of Chemistry and Pharmaceutical Sciences,Qingdao Agricultural University,Qingdao 266109;Chongqing Key Laboratory of Natural Product Synthesis and Drug Research,Innovative Drug Research Center,School of Pharmaceutical Sciences,Chongqing University,Chongqing 401331)
出处
《有机化学》
SCIE
CAS
CSCD
北大核心
2024年第5期1667-1674,共8页
Chinese Journal of Organic Chemistry
基金
国家自然科学基金(No.21772107)
山东省高等学校青创人才引育计划(2021)资助项目。