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微波诱导合成5-芳氧亚甲基-2-[5′-(4″-氯代苯基)-2′-呋喃甲酰胺基]-1,3,4-噁二唑 被引量：1

Microwave induced synthesis of 5-aryloxymethylene-2-[5′-(4″- chlorophenyl)-2′-furoylamido]-1,3,4-oxadiazoles
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摘要 在微波辐射条件下,由1 芳氧乙酰基 4 [5′ (4″ 氯代苯基) 2′ 呋喃甲酰基]氨基硫脲(1a～1i)在醋酸汞存在下,快速环合合成了一系列5 芳氧亚甲基 2 [5′ (4″ 氯代苯基) 2′ 呋喃甲酰胺基] 1,3,4 二唑(2a～2i). aryloxymethylene 2 [5′ (4″ chlorophenyl) 2′ furoylamido] 1,3,4 oxadiazoles(2a～2i) are rapidly synthesized under microwave irradiation by the cyclization of 1 aryloxyacetyl 4 [5′ (4″ chlorophenyl) 2′ furoyl] thiosemicarbazides(1a～1i) in the presence of mercuric acetate.
作者 杨靖亚 王俊科 李政 王喜存
机构地区 西北师范大学化学化工学院
出处 《西北师范大学学报（自然科学版）》 CAS 2003年第3期51-53,共3页 Journal of Northwest Normal University(Natural Science)
基金 甘肃省自然科学基金资助项目(ZS021 A25 006 Z) 甘肃省环保基金资助项目(GH2002 16) 西北师范大学科技创新工程资助项目(NWNU KJCXGC 02 08)
关键词 1 3 4-噁二唑 氨基硫脲 微波辐射 oxadiazole thiosemicarbazide microwave irradiation
分类号 O621.392 [理学—有机化学]
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参考文献13

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同被引文献12

  • 1王喜存,刘娟,李政.微波辐射条件下合成2-芳基-5-[5′-(4″-氯代苯基)-2′-呋喃基]-1,3,4-噁二唑[J].西北师范大学学报（自然科学版）,2004,40(4):49-51. 被引量：1
  • 2张自义,陈立民,冯小明,曾福礼.酰氨基硫脲及其相关杂环衍生物的研究——Ⅻ.1-(α-苯基氰乙酰胺基)-3-芳酰基硫脲及3-(α-苯基氰甲基)-4-芳酰基-1,2,4-三唑-5-硫酚衍生物的合成[J].有机化学,1989,9(2):150-155. 被引量：16
  • 3OZNUR A, AYSE K, NESRIN C, GULTEN O. Synthesis and antimicrobial activity of some 5-aryl-2- [-(N, N-disubstituted thiocarbamoylthio) acylamino] -1,3,4-oxadiazole[J]. Farmaco, 1998, 53: 541- 544.
  • 4ERHAN P, GULAY S, PELIN K. Synthesis and anti- inflammatory activity of 1 - acylthiosemi - carbazides, 1,3,4 - oxadiazoles, 1,3,4 - thiadiazoles and 1,2,4-triazole-3-thiones[J]. Farmaco, 2002, 57: 101-107.
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西北师范大学学报（自然科学版）
2003年 第3期

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