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3-氨基-2-羟基-4-苯基丁酸合成路线图解

Graphical Synthetic Routes of 3-Amino-2-hydroxy-4-phenylbutyric Acid
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作者 张震 徐文方
机构地区 山东大学药学院药物化学研究所
出处 《中国医药工业杂志》 CAS CSCD 北大核心 2003年第11期590-592,共3页 Chinese Journal of Pharmaceuticals
关键词 3-氨基-2-羟基-4-苯基丁酸 合成路线 非天然氨基酸 苯丙氨酸法 天冬氨酸法
分类号 R977.4 [医药卫生—药品]
  • 相关文献

参考文献23

  • 1藤井正 柳内浩司.3-Nitro-2-hydroxy-4-phenylbutyric acids[P].JP:56108743.1981—08—28.
  • 2汝奇,木村徹,木曾良明.立体选择性合成（2S，3S）－3－氨基－2－羟基－4－苯基丁酸[J].中国医药工业杂志,1994,25(12):557-559. 被引量：2
  • 3徐文方,郁有农,张世军,袁玉梅.2-羟基-3-氨基-4-苯丁酸的合成[J].中国医药工业杂志,2001,32(2):79-81. 被引量：5
  • 4Suda H, Takita T, Aoyagi T, et al. The structure of bestatin[J], J Antibiot, 1976,29(1) :100-101.
  • 5Mimoto T, Imai J, Kisanuki S, et al. Kynostatin (KNI)-227 and -272, highly potent anti-HIV agents:conformationally constrained tripeptide inhibitors of HIV protease containing allophenylnorstatine[J].Chem Pharm Bull,1992,40(8):2251-2253.
  • 6Iizuka K, Kamijo T, Harada H, et al. Design and synthesis of an orally potent human renin inhibitor containing a novel amino acid, cyclohexylnorstatines[J ]. J Chem Soc , Chem Commun , 1989, (21): 1678-1680.
  • 7Nishizawa R, Saino T, Takita T, et al. Synthesis and structure-activity relations of hestatin analogs,inhibitors of aminopeptidase B[J]. J Med Chem,1977,20(4) :510-515.
  • 8Fuyuhik M, Teruyo M, Masako O. A practical synthesis of threo-3-amino-2-hydroxy earboxylie acids[J ]. Bull Chem Soc Jpn, 1992,65 : 360- 365.
  • 9Baenziger M, Warm A, Megarrity J. Process for the preparation of a-hydroxy-β-amino carboxylic acid[P]. EP: 543343, 1993-05-26. (CA 1993, 119:160824a).
  • 10Matsumoto S, Matsuo K, Sugawa T. Process for preparing β-amino-a-hydroxy acid derivatives [P].WO : 9807687,1998-02-26. (CA 1998,128: 205135f).

二级参考文献10

  • 1Nishzawa R,Tesushi S,Masao S.A facile synthesis of bestatin[].Journal of Antibiotics.1983
  • 2Fuyuhik M,Teruyo M,Masako O.A practical synthesis of threo-3-amino-2-hydroxycarboxylic acids[].Bulletin of the Chemical Society of Japan.1992
  • 3Hayashi S,Yasohara Y,Yoshihiko H.Method for producing 2-hydroxy-3-nitro-3-butenoic acid and 3-amino-2-hydroxybutanoic acid derivatives[].JP:.1995
  • 4Worrall DE.-Nitro-styrenes[].Org Syn coll vol.1948
  • 5Yuko K,Yoshiji T,Yoshio I.A novel synthesis of the (2R,3S )-and (2R, 3R)-3-amino-2-hydroxycarboxylic acid derivatives, the key components of arenin inhibitor and bestatin,from methyl ( R )-and ( S )-mandelate[].Tetrahedron Letters.1990
  • 6Herranz R,Castro-Pichel J,Vinuesa S.An improved one-pot method for the stereoselective synthesis of the ( 2S , 3R )-3amino-2-hydroxy acids, key intermediates for bestatin and amastatin[].Journal of Organic Chemistry.1990
  • 7Achintya K,Sinhabab U,Ronald T.Silica gel -assisted reduction of nitrostyrenes to 2-aryl -1-nitroalkanes with sodium borohydride[].Tetrahedron Letters.1983
  • 8Suda H,Takita T,Aoyagi T.The structure of bestatin[].Journal of Antibiotics.1976
  • 9Suda H,Takita T,Aoyagi T.The chemical synthesis of bestatin[].Journal of Antibiotics.1976
  • 10Bryan H,Michelle L,Takeo K.A stereospecific synthesis of(-)-bestatin from L-malic acid[].Tetrahedron Letters.1992

共引文献5

中国医药工业杂志
2003年 第11期

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