A direct C–H amination reaction of N-Ts-2-Styrylaniline derivatives to realize the synthesis of indole derivatives was developed in the presence of copper salt. A variety of N-Ts-2-Styrylaniline derivatives were tran...A direct C–H amination reaction of N-Ts-2-Styrylaniline derivatives to realize the synthesis of indole derivatives was developed in the presence of copper salt. A variety of N-Ts-2-Styrylaniline derivatives were transformed into the corresponding indole products in good to excellent yield under mild conditions with the oxidation of potassium persulfate.展开更多
基金financially supported by the National Natural Science Foundation of China(Nos.21272169,21302135)the Key Innovation Team of Science & Technology in Zhejiang Province(No.2010R50018-10)+1 种基金the Science and Technology Bureau of Taizhou(No.08KY10)the Key Disciplines of Applied Chemistry of Zhejiang Province,Taizhou University
文摘A direct C–H amination reaction of N-Ts-2-Styrylaniline derivatives to realize the synthesis of indole derivatives was developed in the presence of copper salt. A variety of N-Ts-2-Styrylaniline derivatives were transformed into the corresponding indole products in good to excellent yield under mild conditions with the oxidation of potassium persulfate.
