A novel route for the synthesis of thiazolo[3,2-a]pyrimidin-7-ones and pyrido[1,2-a]pyrimidin-2,ones from acetylated 2- aminothiazoles and 2-aminopyridines under Vilsmeier conditions has been developed. The plausible ...A novel route for the synthesis of thiazolo[3,2-a]pyrimidin-7-ones and pyrido[1,2-a]pyrimidin-2,ones from acetylated 2- aminothiazoles and 2-aminopyridines under Vilsmeier conditions has been developed. The plausible mechanism has also been proposed.展开更多
基金Zhejiang Key Innovation Team of Green Pharmaceutical Technology (Project No.:2012R20043-12)
文摘A novel route for the synthesis of thiazolo[3,2-a]pyrimidin-7-ones and pyrido[1,2-a]pyrimidin-2,ones from acetylated 2- aminothiazoles and 2-aminopyridines under Vilsmeier conditions has been developed. The plausible mechanism has also been proposed.
