OPIOID δ RECEPTOR IRREVERSIBLE INHIBITORS 2.SYNTHESIS OF ISOTHIOCYANATE DERIVATIVES OF CARFENTANIL AND 4-METHOXYMETHYLFENTANYL

Abstract: The synthesis of isothiocyanate derivatives of carfentanil and 4-methoxymethyl-fentanyl was described.

OPIOID δ RECEOTIR IRREVERSIBLE INHIBITORS 3.SYNTHESIS OF AMIDE ANALOGHES OF SUPERFIT CARFIT AND METHOFIT

Abstract: The Synthesis of 2-furancarboxamide, 2-thiopllenecarboxamide and 2tetrahydro-furancarboxa mide analogues of SuperFIT, CarFIT and MethoFIT was described.

OPIOID & RECEPTOR IRREVERSIBLE INHIBITORS 1.SYNTHESIS AND ABSOLUTE CONFIGURATION OF OHMEFENTANYL ISOTHIOCYANATE ENANTIOMERS

Abstract: The Synthesis of eight enantiomers of ohmefentanyl isothiocyanate and the determination of their absolute configuration were described.